Publications in 2023
Publications are the primary method for reporting and long-term documentation of the research conducted at the NIPER-Hyderabad. Here the list of publications published in year wise...
- Vaibhavi Srivastava , Padakanti Sandeep Chary , Naveen Rajana , Ekta R. Pardhi , Vivek Singh, Dharmendra Khatri , Shashi Bala Singh, Neelesh Kumar Mehra*. Complex ophthalmic formulation technologies: Advancement and future perspectives. J Drug Deliv Sci Technol. 2023. 104317, doi:https://doi.org/10.1016/j.jddst.2023.104317. (Impact factor 5.062).
- 2. Safiya Sulthana, Padakanti Sandeep Chary, Valamala Bhavana, Ekta Pardhi, Shashi Bala Singh, Neelesh Kumar Mehra.* Development and evaluation of emulgel for Effective Management of the Imiquimod Induced Psoriasis. Inflammopharmacology. 2023 Jan 7. doi: 10.1007/s10787-022-01131-7 (Impact Factor 5.0093).
- Purva Pingle, Atul Mourya, Madhulika Namdeo, Katta Chanti Babu, Harithasree Veerabomma, Radheshyam Maurya, Pankaj Kumar Singh, Neelesh Kumar Mehra, Saurabh Srivastava, Jitender Madan. Andrographolide-Soya-L-α-phosphatidyl choline complex augmented solubility and drug delivery in Leishmania donovani, a causative agent for cutaneous and visceral leishmaniasis. AAPS PharmSciTech. 2023 24(1):46. doi: 10.1208/s12249-023-02507 (Impact factor 4.026).
- Arti Mehndole, Nitita Walke, Srusti Mahajan, Mayur Alhare, Indrani Maji, Ujala Gupta, Neelesh Kumar Mehra, Pankaj Kumar Singh. Core-shell type lipid and polymeric nanocapsules: The Transformative Multifaceted Delivery System. AAPS PharmSciTech. 2023 in press, (Impact factor 4.026).
- Pratik Kharat, Padakanti Sandeep Chary, Naveen Rajana, Valamla Bhavana, Geetanjali, Chandraiah Godugu, Shashi Bala Singh, Neelesh Kumar Mehra*. Thymoquinone Loaded Essential Oil Based Emulgel as an armament for Anti-psoriatic Activity. AAPS PharmSciTech. 2022; 24: 26. (Impact factor 4.026). doi 10.1208/s12249-022-02482-8.
- S. Kumar, S. Nunewar, Kanchupalli, V.* “Rh (III)‐Catalyzed Cross‐Coupling/Annulation of Two Carbene Precursors: Construction of Dihydrobenzo [c] chromen‐6‐one Scaffolds and Application in the Total Synthesis of Cannabinol” (doi.org/10.1002/ajoc.202100689) Asian. J. Org. Chem. 2022, 11, e202100689 (Selected for Hot topic). (IF 3.3)
- S. Kumar, S. Nunewar, T. Sabbi, Kanchupalli, V.* “Synthesis of Indenone Derivatives by Rh(III)-Catalyzed C-H Functionalization of Sulfoxonium Ylides with 1,3-Diynes” Org. Lett. 2022, 24, 3395–3400. (doi.org/10.1021/acs.orglett.2c01166) (IF 6.02)
- S. Nunewar, S. Kumar, H. Pendam P., Pradeep G., Kanchupalli, V.* “Solvent Controlled Rh(III)-Catalyzed Switchable [4+2] Annulation of 2-ArylIndoles with Iodonium Ylides” Chem. Commun., 2022, 58, 6140-6143. (doi.org/10.1039/D2CC01386J) (IF 6.3)
- S. Nunewar, S. Kumar, A. W. Meshram, Kanchupalli, V.* “Ru(II)-Catalyzed C−H Functionalization of 2-Arylbenzimidazoles with Iodonium Ylides: A straightforward access to bridgehead Polycyclic N-Heterocycles” J. Org. Chem. 2022, 87, 13757–13762 (doi.org/10.1021/acs.joc.2c01429) (IF 4.2).
- S. Kumar, T. Sabbi, Pradeep, G., Rasika. P., Kanchupalli, V.* “1,3-Diynes: A Versatile Precursor in Transition-Metal Catalyzed (Mediated) C-H Functionalizations:” Chem. Rec., 2022 (DOI: 10.1002/tcr.202200228) (IF 6.9).
- Kanchupalli, V.; Kalepu, J.; Joseph, D.; Arshad, M.; Thorbole, L.; Katukojvala, S. “Rhodium-Catalyzed Enal-Transfer with N-Methoxypyridazinium Salts” Org. Lett. 2022, 24, 3850–3854. (doi.org/10.1021/acs.orglett.2c01424) (IF 6.02)
- S. Kumar, V. Borkar, M. Mujahid, S. Nunewar, Kanchupalli, V.* “Iodonium Ylides: An emerging and alternative carbene precursor for C-H functionalizations:” Org. Biomol. Chem., 2023, 21, 24-38 (doi.org/10.1039/D2OB01644C) (IF 3.89).
- Kumar, S, V. Borkar, S. Nunewar, S. Yadav, Kanchupalli, V.* “Rh(III)-Catalyzed C−H Annulation of Sulfoxonium Ylides and 1,3-Diynes: A Rapid Access to Alkynyl-1-Naphthol Derivatives” Chem Asian J. (Just accepted). (IF 4.8).
- Gautam Kumar and Asha Kiran Tudu: Tackling multidrug-resistant Staphylococcus aureus by natural products and their analogues acting as NorA efflux pump inhibitors. Bioorg. Med. Chem. 80 (2023) 117187. IF: 3.41
- Gautam Kumar and Shobhna Kapoor: Targeting Mycobacterial Membranes and Membrane Proteins: Progress and Limitations. https://doi.org/10.1016/j.bmc.2023.117212. IF: 3.41
- Synthesis and cytotoxicity evaluation of DNA-interactive β-carboline indolyl-3-glyoxamide derivatives: Topo-II inhibition and in silico modelling studies; Soni, J. P.; Reddy, G. N.; Rahman, Z.; Sharma, A.; Spandana, A.; Phanindranath, R.; Dandekar, M. P.; Nagesh, N.;Shankaraiah, Bioorg. Chem., 2023, 131, 106313
- A tribute to Professor Ahmed Kamal (AK-1494BT); Shankaraiah, N. Arkivoc 2023, iii, 1-9
- Development of hydrazide hydrazone-tethered combretastatin-oxindole derivatives as antimitotic agents; Bora, D.; Sharma, A.; John, S. E.; Shankaraiah, N. J. Mol. Str., 2023, 1275, 134675
- Benzimidazole based bis-carboxamide derivatives as promising cytotoxic agents: Design, synthesis, in silico and tubulin polymerization inhibition; Laxmikeshav, K.; Sharma, P.; Palepu, M.; Sharma, P.; Mahale, A.; George, J.; Phanindranath, R.; Dandekar, M. P.; Kulkarni, O.P.; Nagesh, N.; Shankaraiah, N. J. Mol. Str., 2023, 1271, 134078
In Press
- Design, synthesis and in vitro cytotoxicity evaluation of indolo-pyrazoles grafted with thiazolidinone as tubulin polymerization inhibitors; Soni, J. P.; Chilvery, S.; Sharma, A.; Reddy, G. N.; Godugu, C.; Shankaraiah, N. RSC Med. Chem., 2023
- Exploration of cytotoxic potential and tubulin polymerization inhibition activity of cis-stilbene-1,2,3-triazole congeners; Bora, D.; Samir, K. M.; Sharma, A.; Chilvery, S.; Bansod, S.; John, S. E.; Godugu, C.; Shankaraiah, N. RSC Med. Chem., 2023
- Synthesis of cis-stilbene based 1,2,4-triazole/1,3,4-oxadiazole conjugates as potential cytotoxic and tubulin polymerization inhibitors; John, S. E.; Sharma, A.; Gulati, S.; Bora, D.; Shankaraiah, N. New. J. Chem., 2023
- 1,2,3-Triazolo-2-aryl-linked benzimidazole derivatives as tubulin polymerization inhibitors and DNA intercalators: Design, synthesis, biological evaluation and docking studies; Laxmikeshav, K.; Sayali, M.; Devabattula, G.; Sharma, P.; Mahale, A.; George, J.;Phanindranath, R.; Godugu, C.; Kulkarni, O. P.; Nagesh, N.; Shankaraiah, N. Archiv der Pharmazie 2023