Publications in 2016
Publications are the primary method for reporting and long-term documentation of the research conducted at the NIPER-Hyderabad. Here the list of publications published in year wise...
- Nagula Shankaraiah, Chetna Jadala, Shalini Nekkanti, Kishna Ram Senwar, Narayana Nagesh, Shweta Shrivastava, VGM Naidu, Manda Sathish, Ahmed Kamal; Design and synthesis of C3-tethered 1, 2, 3-triazolo-β-carboline derivatives: Anticancer activity, DNA-binding ability, viscosity and molecular modeling studies. Bioorganic chemistry, 2016, 64, 42-50.
- Lalita Guntuku, VGM Naidu, Veera G Yerra.; Mitochondrial Dysfunction in Gliomas: Pharmacotherapeutic Potential of Natural Compounds. Current neuropharmacology 2016, 14(6),567-583
- Kishna Ram Senwar, T Srinivasa Reddy, Dinesh Thummuri, Pankaj Sharma, VGM Naidu, Gannoju Srinivasulu, Nagula Shankaraiah.; Design, synthesis and apoptosis inducing effect of novel (Z)-3-(3′-methoxy-4′-(2-amino-2-oxoethoxy)-benzylidene) indolin-2-ones as potential antitumour agents. European journal of medicinal chemistry, 2016, 118, 34-46.
- Kishna Ram Senwar, T Srinivasa Reddy, Dinesh Thummuri, Pankaj Sharma, Suresh K Bharghava, VGM Naidu, Nagula Shankaraiah.;Design and synthesis of 4′-O-alkylamino-tethered-benzylideneindolin-2-ones as potent cytotoxic and apoptosis inducing agents. Bioorganic & Medicinal Chemistry Letters, 2016, 26(16), 4061-4069.
- Pankaj Sharma, Dinesh Thummuri, T Srinivasa Reddy, Kishna Ram Senwar, VGM Naidu, Gannoju Srinivasulu, Suresh K Bharghava, Nagula Shankaraiah.; New (E)-1-alkyl-1H-benzo [d] imidazol-2-yl) methylene) indolin-2-ones: Synthesis, in vitro cytotoxicity evaluation and apoptosis inducing studies. European Journal of Medicinal Chemistry, 2016 , 122, 584-600.
- Pankaj Sharma, T Srinivasa Reddy, Dinesh Thummuri, Kishna Ram Senwar, Niggula Praveen Kumar, VGM Naidu, Suresh K Bhargava, Nagula Shankaraiah.; Synthesis and biological evaluation of new benzimidazole-thiazolidinedione hybrids as potential cytotoxic and apoptosis inducing agents. European Journal of Medicinal Chemistry, 2016, 124, 608-621.
- Uttam B. Karale, Saradhi Kalari, Jala Shivakumar, Vitthal B. Makane, Dattatraya A. Babar, Ritesh P. Thakare, Bathini Nagendra Babu, Sidharth Chopra, Haridas B. Rode*.; Ligand-free Pd-catalysed decarboxylative arylation of imidazo[1,2-a]pyridine-3-carboxylic acids with aryl bromides. RSC Adv., 2016, 6, 65095–65104.
- K. N. Visweswara Sastry, Sunitha Rani Routhu, Soma Gupta Datta, Narayana Nagesh, Bathini Nagendra Babu, Jagadeesh Babu Nanubolu, C. Ganesh Kumar, Ram Awatar Maurya*, Ahmed Kamal*.; Synthesis, DNA binding affinity and anticancer activity of novel 4H-benzo[g][1,2,3]triazolo[5,1-c] [1,4]oxazocines. Org. Biomol. Chem., 2016, 14, 9294–9305.
- Atulya Nagarsenkar, Lalita Guntuku, Sravanthi Devi Guggilapu, Danthi Bai K., Srinivasulu Gannoju, V.G.M. Naidu,**, Nagendra Babu Bathini.*; Synthesis and apoptosis inducing studies of triazole linked 3-benzylidene isatin derivatives. European Journal of Medicinal Chemistry, 2016, 124, 782-793.
- Rahul B, Chavan, Rajesh Thipparaboina, Dinesh Kumar and Nalini R. Shastri.; Co amorphous systems: A product development perspective. Int. J. Pharm, 2016, 515, 403–415.
- Anjali Jain, Konda Reddy Kunduru, Arijit Basu, Boaz Mizrahi, Abraham J. Domb, Wahid Khan.; Injectable formulations of poly(lactic acid) and its copolymers in clinical use. Adv. Drug Deliv. Rev, 2016, 107, 213–227.
- Arijit Basu, Konda Reddy Kunduru, Sindhu Doppalapudi, Abraham J. Domb, Wahid Khan, Poly(lactic acid) based hydrogels. Adv. Drug Deliv. Rev, 2016, 107, 2016, 192–205.
- Anjali Jain, Sindhu Doppalapudi, Abraham J. Domb, Wahid Khan.; Tacrolimus and curcumin co-loaded liposphere gel: Synergistic combination towards management of psoriasis. J. Control. Release, 2016, 243, 132–145.
- Sameer S. Katiyar, Eameema Muntimadugu, Towseef Amin Rafeeqi, Abraham J. Domb, Wahid Khan.; Co-delivery of rapamycin and piperine loaded polymeric nanoparticles for breast cancer treatment. Drug Deliv., 2016, 23, 2608-2616.
- Diana E. Ickowicz, Ester Abtew, Wahid Khan, Ludmila Golovanevski, Carolyn F. Weiniger,Abraham J. Domb.; Poly(ester-anhydride) for controlled delivery of hydrophilic drugs. J. Bioact. Compat. Pol., 2016, 31, 127-139.
- Sindhu Doppalapudi, Anjali Jain, Upendra Bulbake, Wahid Khan.; Nanotherapeutics: Emerging trends in management of psoriasis. Pharm Nanotechnol. 2016, 4, 1-17.
- Rohan Ghadi, Eameema Muntimadugu, A.J. Domb, Wahid Khan, Xiang Zhang., Synthetic biodegradable medical polymer: Polyanhydrides, Science and Principles of Biodegradable and Bioresorbable Medical Polymers Eds: Xiang Zhang. Elsevier Publications 2016, 153-187.
- Naveen Chella, Bhaskar Daravath, Dinesh Kumar, Rama Rao Tadikonda.; Formulation and Pharmacokinetic Evaluation of Polymeric Dispersions Containing Valsartan. European Journal of Drug Metabolism and Pharmacokinetics. 2016, 41(5), 517–526.
- P Komirishetti, A Areti, R Gogoi, R Sistla, A Kumar.; PARP inhibition reveals a potential mechanism to promote neuroprotection and for the treatment of neuropathic pain. Neural Regeneration Research, 2016, 11 (10), 1545-1548.
- S Reddemma, VG Yerra, P Komirishetty, A Areti, A Kumar.; Fisetin Imparts Neuroprotection in Experimental Diabetic Neuropathy by Modulating Nrf2 and NF-κB Pathways. Cellular and Molecular Neurobiology, 2016, 36 (6), 883-892.
- N. Satheeshkumar, David Paul, A. Lingesh.; Liquid Chromatography-Mass Spectrometry (LC-MS) - Approaches to Adulterant Detection in Herbal Products. Tsay, H.-S., Shyur, L.-F., Agrawal, D.C., Wu, Y.-C., Wang, S.-Y. (Eds.) Medicinal Plants - Recent Advances in Research and Development. Springer International Publishing, Switzerland , 2016, 73-95.
- N. Satheeshkumar, R.S. K Vijayan, A. Lingesh, S. Santhikumar and Ch. Vishnuvardhan.; Spices: Potential Therapeutics for Alzheimer’s Disease. M.M. Essa et al. (eds.), The Benefits of Natural Products for Neurodegenerative Diseases, Advances in Neurobiology. Springer International Publishing Switzerland, 2016, 12, 57-78.
- Chiguru Vishnuvardhan , Debasish Swain , Roshan Borkar , S. Gananadhamu , R. Srinivas , N. Satheeshkumar.; Study of forced degradation behaviour of brinzolamide using LC-ESI- Q-TOF and in silico toxicity prediction. Chromatographia, 2016, 79, 1293.
- Senwar, K. R.; Sharma, P.; Reddy, T. S.; Thummuri, D.; Naidu, V.G.M.; Shankaraiah, N.; Design, synthesis and apoptosis inducing novel (Z)-3-(3'-methoxy-4'-(2-amino-2-oxoethoxy)-benzylidene)indolin-2-ones as potential cytotoxic agents. Eur. J. Med. Chem., 2016, 118, 34–46.
- Shankaraiah, N.; Sharma, P.; Pedapati, S.; Nekkanti, S.; Srinivasulu, V.; Kumar, N. P.; Kamal, A.; Synthesis of Novel C3-Linked β-Carboline-Pyridine Derivatives Employing Khronke Reaction: DNA-binding Ability and Molecular Modeling Studies. Lett. in Drug Design & Discovery, 2016, 13, 335–342.
- Manish Kumar Jeengar.; Sri Vishnu Kiran Rompicharla.; Shweta Shrivastava.; Naveen Chella.; Nalini R Shastri.; VGM Naidu.; Ramakrishna Sistla.; Emu oil based nano-emulgel for topical delivery of curcumin. International journal of pharmaceutics, 2016, 506, 222-236.
- Rajesh Kumar Gurram.; Suchithra Gandra.; Nalini R Shastri.; Design and optimization of disintegrating pellets of MCC by non-aqueous extrusion process using statistical tools. Eur J Pharm Sci., 2016, 84, 146–156.
- Amitha Thakur.; Rajesh Thipparaboina.; Dinesh Kumar.; Kodukula Sai Gouthami.; Nalini R Shastri.; Crystal Engineered Albendazole with Improved Dissolution and Material Attributes. CrystEngComm, 2016, 18, 1489-1494.
- Rajesh Thipparaboina.; Dinesh Kumar.; Rahul B. Chavan.; Nalini R. Shastri.; Multidrug co-crystals: towards the development of effective therapeutic hybrids. Drug Discov Today, 2016, 21, 481–490.
- Supriya Dattatray Jitkar.; Rajesh Thipparaboina.; Rahul B Chavan.; Nalini R. Shastri.; Spherical Agglomeration of Platy Crystals: Curious Case of Etodolac. Cryst. Growth Des, 2016, 16, 4034–4042.
- Rajesh Thipparaboina.; Sudhir Mittapalli.; Sowjanya Thatikonda.; Ashwini Nangia.; V. G. M. Naidu.; and Nalini R Shastri.; Syringic Acid: Structural Elucidation and Co-Crystallization. Cryst. Growth Des., 2016, 16, 4679–4687.
- Rahul B. Chavan.; Rajesh Thipparaboina.; Dinesh Kumar.; Nalini R. Shastri.; Evaluation of the inhibitory potential of HPMC, PVP and HPC polymers on nucleation and crystal growth. RSC Adv., 2016, 6, 77569.
- Prinesh N. Patel.; Pradipbhai D. Kalariya.; Swamy C.V.; Gananadhamu S.; Srinivas R.; Quantitation of acotiamide in rat plasma by UHPLC-Q-TOF-MS: method development, validation and application to pharmacokinetics. Biomed Chromatogr, 2016, 30, 363-368.
- Debasish Swain.; Prinesh N Patel.; Gangam Nagaraj.; Kona S Srinivas.; Mahesh Sharma.; Prabha Garg.; Gananadhamu Samanthula.; Liquid Chromatographic Method Development for Forced Degradation Products of Dabigatran Etexilate: Characterisation and In Silico Toxicity Evaluation. Chromatographia, 2016, 79, 169-178.
- Debasish Swain.; Gananadhamu Samanthula.; Shweta Bhagat.; P.V. Bharatam.; Venkatakrishna Akula.; Barij N. Sinha.; Characterization of forced degradation products and in silico toxicity prediction of Sofosbuvir: A novel HCV NS5B polymerase inhibitor. J. Pharm. Biomed. Anal., 2016, 120, 352-363.
- Talluri* M.V.N.K.; Kalariya, P.D.; Dharavath. S,; Automated statistical experimental design approach for rapid separation of coenzyme Q10 and its biotechnological process related impurities using UPLC and UPLC/APCI/MS. J Sep Sci., 2016 39(18), 3528-35.
- Mahamuni. B. S, Jajula. A, Awasthi A, Kalariya. P. D, Talluri, M.V.N.K.; Selective separation and characterisation of stress degradationproducts and process impurities of prucalopride succinate by LC-QTOF-MS/MS. J. Pharm. Biomed. Anal, 2016, 125, 219–228.
- Uttam B. Karalea, Saradhi Kalaria, Jala Shivakumar, Vitthal B. Makanea, Dattatraya A. Babara, Ritesh P. Thakare, Bathini Nagendra Babu, Sidharth Chopra, Haridas B. Rode,; Ligand-free Pd-catalysed decarboxylative arylation of Imidazo[1,2-a]pyridine-3-carboxylic acids with Aryl bromides. RSC Advances, 2016 , 69.
- Atulya N., S. K. Prajapti, Sravanthi Devi G., Swetha B., Sudha S. K., Ramesh U., Bathini Nagendra Babu,; Investigation of triazole-linked indole and oxindole glycoconjugates as potential anticancer agents: novel Akt/PKB signaling pathway inhibitors. RSC, MedChemComm, 2016 7, 646.
- S. K. Prajapti, Atulya N., Sravanthi Devi G., Gupta, K., Lingesh A, Manish Kumar J., V. G. M. Naidu, Bathini Nagendra Babu,; Synthesis and biological evaluation of oxindole linked indolyl-pyrimidine derivatives as potential cytotoxic agents. Bioorganic & Medicinal Chemistry Letters, 201626, 3024.
- Sravanthi Devi G., S. K. Prajapti, Atulya N., G. Lalita, V.G.M. Naidu and Bathini Nagendra Babu.; MoO2Cl2 catalyzed efficient synthesis of functionalized 3,4-dihydropyrimidin-2(1H)-ones / thiones and polyhydroquinolines: Recyclability, Fluoroscence and Biological studies. RSC New Journal Chemistry, 2016, 40, 838.
- Sravanthi Devi G, S. K. Prajapti, Atulya N, Keshav K. G., Bathini Nagendra Babu.; Indium(III) Chloride Catalyzed Synthesis of 5-Substituted 1H-Tetrazoles from Oximes and Sodium Azide. Synlett, 2016, 27, 1241.
- Bandaru, S.; Alvala, M.; Akka, J.; Sagurthi, S. R.; Nayarisseri, A.; Singh, S. K.; Mundluru, H. P., Identification of Small Molecule as a High Affinity beta2 Agonist Irrespectively Targeting Wild and Mutated (Thr164Ile) beta 2 Adrenergic Receptor in the Treatment of Bronchial Asthma. Current pharmaceutical design, 2016.
- Narva, S.; Chitti, S.; Bala, B. R.; Alvala, M.; Jain, N.; Kondapalli, V. G.; Synthesis and biological evaluation of pyrrolo[2,3-b]pyridine analogues as antiproliferative agents and their interaction with calf thymus DNA. European journal of medicinal chemistry, 2016, 114, 220-31.
- Muntimadugu, E.; Dhommati, R, Jain, A.; Challa, V.G.S.; Shaheen, M.; Khan, W.; Intranasal delivery of nanoparticle encapsulated tarenflurbil: A potential brain targeting strategy for Alzheimer’s disease. Eur. J. Pharm. Sci. 2016, 92, 224-234.
- Muntimadugu, E.; Kumar, R.; Saladi, S.; Rafeeqi, T.A.; Khan, W.; CD44 targeted chemotherapy for co-eradication of breast cancer stem cells and cancer cells using polymeric nanoparticles of salinomycin and paclitaxel. Colloids Surf., B. 2016, 143, 532-546.
- Doppalapudi, S.; Jain A.; Domb, A.J.; Khan, W.; Biodegradable polymers for targeted delivery of anticancer drugs; Expet Opin. Drug Deliv. 2016, 13(6) 891-909.
- Singh, I.; Swami, R.; Pooja, D.; Jeengar, M.K.; Khan, W.; Ramakrishna, S.; Lactoferrin Bioconjugated Solid Lipid Nanoparticles: A New Drug Delivery System for Potential Brain Targeting. J. Drug Target. 2016, 24(3), 212-23.
- Singh, I.; Swami, R.; Khan, W.; Ramakrishna, S.; Chapter 11, Lymphatic System: A Prospective Area for Advanced Targeting of Particulate Drug Carriers. Handbook of Immunological Properties of Engineered Nanomaterials. World Scientific Publishing, 2016, 2, 363-398.
- Basu, A.; Farah, S.; Kunduru K.R.; Doppalapudi, S.; Khan W.; Domb A.J.; Chapter 8, Polyurethanes for controlled drug delivery, Advances in Polyurethane Biomaterials, Eds: Cooper & Guan. 1st Edition, Elsevier Publications, 2016, 217-246.
- Ghadi, R.; Jain, A.; Khan, W.; Domb, A. J.; Chapter 12, Microparticulate polymers and hydrogels for wound healing, Wound Healing Biomaterials - Volume 2: Functional Biomaterials Eds: Magnus Agren. Elsevier Publications, 2016, 203-225.
- Kommineni, N.; Khan, W.; Nanomedicine in global market; Nano Digest, July 2016, 36-41.
- Vishnuvardhan Ch, Allakonda L, Srinivas R, Satheeshkumar N.; Forced degradation study of racecadotril: Effect of co-solvent, characterization of degradation products by UHPLC-Q-TOF-MS/MS, NMR and cytotoxicity assay. Journal of Pharmaceutical and Biomedical Analysis, 2016, 128, 9–17.
- Chiguru Vishnuvardhan , Saibaba Baikadi, Roshan M Borkar, R. Srinivas, N. Satheeshkumar.; In vivo metabolic investigation of silodosin using UHPLC–QTOF–MS/MS and in silico toxicological screening of its metabolites. Journal of Mass Spectrometry, 2016.
- Syed Safiullah Ghori, Md Ikram Ahmed, Md. Arifuddin, Md Shoaibuddin Khateeb.; Evaluation of analgesic and anti-inflammatory activities of formulation containing camphor, menthol and thymol. International Journal of Pharmacy and Pharmaceutical Sciences, 2016, 8 (1), 271-274.
- K. C. Rajanna., Aneesa Ferdose., K. Rajender Reddy., Md. Arifuddin., M. Moaazzam Ali.; Transition metal ions as catalysts for efficient formylation of hydrocarbons with Vilsmeier -Haack reagents: Kinetics and mechanism. Journal of Solution Chemistry, 2016, 45(3), 371-394.
- Safiullah SG, Shazia S, Fouzia F, Ummara H, Arifuddin M, and Tasneem M.; Isolation of Phytosterols from the methanolic extracrt of leaves of Ficus Dalhousiae Miq. RJPBCS, 2016, 7(4), 847-854.
- Nekkanti, S.; Veeramani, K.; Kumar, N. P.; Kamal, A.; Shankaraiah, N.; Microwave-assisted direct oxidative synthesis of α-ketoamides from aryl methyl ketones and amines by a water soluble Cu(I)-complex. Green Chem., 2016, 18, 3439–3447.
- Krishna, N. H.; Saraswati, A. P.; Sathish, M.; Shankaraiah, N.; Kamal, A.; Silver-Catalyzed Domino Aza-Annulation/Diels-Alder Cyclization of 2-ene-yne Anilines: A Facile One-Pot Access to Carbazole, Dihydrocarbazole and Tetrahydrocarbazole Frameworks. Chem. Comm. 2016, 52, 4581–4584.
- Sathish, M.; Chetna, J.; Krishna, N. H.; Shankaraiah, N.; Alarifi, A.; Kamal, A.; Iron-Mediated Concise One-Pot Synthesis of 3, 5-Diarylpyridines from beta-Nitrostyrenes. J. Org. Chem., 2016, 81, 2159–2165.
- Nekkanti, S.; Kumar, N. P.; Sharma, P.; Kamal, A.; Nachtigall, F. M.; Forero-Doria, O.; Santos, L. S.; Shankaraiah, N.; TBAI/TBHP-Catalyzed [3+2] cycloaddition / oxidation / aromatization cascade and online ESI-MS mechanistic studies: Synthesis of pyrrolo[2,1-a]isoquinolines and indolizino[8,7-b]indoles. RSC Adv., 2016, 6, 2671–2677.
- D. Ravikumar Reddy, Amit Khurana, Swarna Bale, Ramu Ravirala, V. Samba Siva Reddy, M. Mohan Kumar, Chandraiah Godugu.; Natural Flavonoids Silymarin and Quercetin Improve the Brain Distribution of Co-administered P-gp Substrate Drugs. SpringerPlus, 2016.
- Swarna Bale, Amit Khurana, Mandip Singh and Chandraiah Godugu.; Overview on Therapeutic Applications of Microparticle Drug Delivery System. Critical Reviews in Therapeutic Drug Carrier Systems, 2016.
- Chandraiah Godugu, Ravi Doddapaneni, Stephen H Safe, Mandip Singh.; Novel Diindolylmethane derivatives based NLC formulations to improve the oral Bioavailability and anticancer effects in Triple Negative Breast Cancer. European Journal of Pharmaceutics and Biopharmaceutics, 2016.
- Srikrishna D, Chandraiah Godugu, Dubey PK.; A Review on Pharmacological properties of Coumarins. 2016.
- Chandraiah Godugu, Singh M.; AlgiMatrix™-Based 3D Cell Culture System as an In Vitro Tumor Model: An Important Tool in Cancer Research. Methods Mol Biol. 2016, 1379,117-28.
- Tiruveedi VL, Bale S, Khurana A, Chandraiah Godugu.; Tankyrase as a Novel Molecular Target in Cancer and Fibrotic Diseases. Curr Drug Targets. 2016.
- Chandraiah Godugu, Doddapaneni R, Patel AR, Singh R, Mercer R, Singh M.; Novel Gefitinib Formulation with Improved Oral Bioavailability in Treatment of A431 Skin Carcinoma. Pharm Res, 2016, 33(1):137-54.
- Sunitha Sampathi, Rakesh Achanta, Pankaj Tiriya, Sonia Gera, P Sravanthi Reddy, Venu Talla.; “Formulation and Evaluation of Carvedilol Loaded Lactide Nanoparticles: An Appraisal to Anti-Hypertensive and Anti-Inflammatory Therapy. Advanced Science, Engineering and Medicine, 2016, 8(7):503-514.
- Sunitha S, Sonia Gera, Srikanth H, Ashok Z.; “Synthesis and evaluation of olmesartan medoxomil complex with SBE7 β-CD for enhanced dissolution and bioavailability”. International Journal of Pharmacy and Pharmaceutical Sciences, 8(1), 2016.
- Jeengar, M., Shrivastava, S., Mouli Veeravalli, S., Naidu, V., and Sistla, R. (2016). Amelioration of FCA induced arthritis on topical application of curcumin in combination with emu oil. Nutrition, 2016, 32: 955-964.
- Kulhari, H., Pooja, D., Shrivastava, S., Kuncha, M., Naidu, V., and Bansal, V. et al. (2016). Trastuzumab-grafted PAMAM dendrimers for the selective delivery of anticancer drugs to HER2-positive breast cancer. Sci. Rep., 2016, 6:23179.
- Areti, A., Yerra, V., Komirishetty, P., and Kumar, A., Potential Therapeutic Benefits of Maintaining Mitochondrial Health in Peripheral Neuropathies. Current Neuropharmacology, 2016, 14(6):593-609.
- Komirishetty, P.; Areti, A.; Sistla, R.; Kumar, A.; Morin Mitigates Chronic Constriction Injury (CCI)-Induced Peripheral Neuropathy by Inhibiting Oxidative Stress Induced PARP Over-Activation and Neuroinflammation. Neurochem Res., 2016, 41(8), 2029-2042.
- Komirishetty, P.; Areti, A.; Yerra, V.; PK, R.; Sharma, S.; Gogoi, R. et al.; PARP inhibition attenuates neuroinflammation and oxidative stress in chronic constriction injury induced peripheral neuropathy. Life Sciences. 2016, 150, 50-60.
- Kumar. A.; Mitochondrial Dysfunction & Neurological Disorders. Current Neuropharmacology. 2016 14(6), 565-566.
- Yerra. V., Gundu. C., Bachewal, P., Kumar. A.; Autophagy: The missing link in diabetic neuropathy?. Medical Hypotheses. 2016 86, 120-128.
- Siresha Bathina.; Nanduri Srinivas.; Undurti N.Das.; BDNF protects pancreatic β cells (RIN5F) against cytotoxic action of alloxan, streptozotocin, doxorubicin and benzo(a)pyrene in vitro; Metabolism, 2016, 65 (5), 667-684.
- Digwal C S, Yadav U, Sakla A P, Ramya P V S, Aaghaz S, Kamal A; VOSO4 catalyzed highly efficient synthesis of benzimidazoles, benzothiazoles, and quinoxalines. Tet. Lett., 57, 2016, 4012.
- Reddy V G, Reddy T S, Nayak V L, Prasad B, Reddy A P, Ravikumar A, Taj S, Kamal A; Design, synthesis and biological evaluation of N-((1-benzyl-1H-1,2,3-triazol-4-yl)methyl)-1,3-diphenyl-1H-pyrazole-4-carboxamides as CDK1/Cdc2 inhibitors. Eur. J. Med. Chem., 2016,122, 164.
- Yellaiah T, Manasa K L, Sathish M, Alarifi A, Kamal A; Phenyliodonium Diacetate Mediated One-Pot Synthesis of Benzimidazoles and Quinazolinones from Benzylamines. Chemistry Select, 2016, 1, 2895.
- Nayak V L, Nagaseshadri B, Vishnuvardhan M V P S, Kamal A; Investigation of the apoptotic pathway induced by benzimidazole–oxindole conjugates against human breast cancer cells MCF-7. Bioorg. Med. Chem. Lett., 2016, 26, 3313.
- Kamal A, Bajee S, Nayak V L, Rao A V S, Nagaraju B, Reddy Ch.R, Kapure J S, Alarifi A; Synthesis and biological evaluation of arylcinnamide linked combretastatin-A4 hybrids as tubulin polymerization inhibitors and apoptosis inducing agents. Bioorg. Med. Chem. Lett., 2016, 26, 2957.
- Srikanth P S, Nayak V L, Babu K S, Kumar G B, Ravikumar A, Kamal A; 2-Anilino-3-Aroylquinolines as Potent Tubulin Polymerization Inhibitors. ChemMedChem, 2016, 11, 2050.
- Kamal A, Nayak V L, Nagesh N, Vishnuvardhan M V P S, Reddy N V S; Benzo[b]furan derivatives induces apoptosis by targeting the PI3K/Akt/mTOR signaling pathway in human breast cancer cells, Bioorganic Chemistry, 2016, 66, 124.
- Borkar R, Bhandi M M, Dubey A P, Reddy V G, Komirishetty P, Nandekar P P, Sangamwar A T, Kamal A, Banerjee S K, Ragampeta S; An Evaluation of the CYP2D6 and CYP3A4 inhibition potential of metoprolol metabolites and their contribution to drug-drug and drug-herb interaction by LC-ESI/MS/MS. Biomedical Chromatography, 2016, 30, 1556.
- Kamal, A; Mahesh, R; Nayak, V.L; Babu, K.S; Kumar, G.B; Shaik, A.B; Kapure, J.S; Alarifi, A; Discovery of pyrrolospirooxindole derivatives as novel cyclin dependent kinase 4 (CDK4) inhibitors by catalyst-free, green approach. Eur. J. Med. Chem., 2016, 108, 476.
- Kamal A, Shaik B, Nayak V L, Rao A V S, Nagaraju B, Reddy Ch R, Kapure J S, Alarifi A; Synthesis and Biological Evaluation of Arylcinnamide linked Combretastatin-A4 hybrids as Tubulin Polymerization Inhibitors and Apoptosis Inducing Agents. Bioorg. Med. Chem. Lett, 2016, 26, 2957.
- Kamal A, Srikanth P S, Vishnuvardhan M V P S, Kumar G B, Babu K S, Hussaini S M A, Kapure J S, Alarifi A. Combretastatin linked 1,3,4-oxadiazole conjugates as a Potent Tubulin Polymerization inhibitors. Bioorganic Chemistry, 2016, 65, 126.
- Suja T D, Divya K V L, Nayak V L, Ravikumar A, Kamal A; Copper-catalyzed three-component synthesis of aminonaphthoquinone–sulfonylamidine conjugates and in vitro evaluation of their antiproliferative activity. Bioorg. Med. Chem. Lett., 2016, 26, 2072.